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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T9855 | BR102910 | 4-Thiazolecarboxamide, N-[2-[(2S)-2-cyano-4,4-difluoro-1-pyrrolidinyl]-2-oxoethyl]-2-[(3,4-dichlorophenyl)methyl]- | Others |
BR102910 (4-Thiazolecarboxamide, N-[2-[(2S)-2-cyano-4,4-difluoro-1-pyrrolidinyl]-2-oxoethyl]-2-[(3,4-dichlorophenyl)methyl]-) is a selective inhibitor of fibroblast activated protein (FAP). | |||
T7890 | SP-13786 | UAMC-1110 | Others |
SP-13786 (UAMC-1110) is an inhibitor of fibroblast activation protein (FAP) (IC50 : 3.2 nM); also inhibits prolyl oligopeptidase (PREP) ( IC50 : 1.8 μM). | |||
T10227 | Ac-Gly-BoroPro | Others | |
Ac-Gly-BoroPro is a selective FAP inhibitor (Ki: 23 nM). | |||
T11264 | FAPI-4 | Others | |
Api-4 is a fibroblast activated protein (FAP) inhibitor used in cancer research. | |||
T78214 | FAP-IN-2 TFA | ||
FAP-IN-2 TFA is a 99mTc-labeled, isonitrile-containing derivative inhibitor of fibroblast activation protein (FAP), utilized for tumor imaging [1]. | |||
T78921 | FAP-IN-1 | ||
FAP-IN-1 is a fibroblast activation protein (FAP) inhibitor, exhibiting an IC50 of 3.3 nM, and is utilized for cancer research [1]. | |||
T74402 | FAP-PI3KI1 | ||
FAP-PI3KI1, a fibroblast-activated protein (FAP)-targeted PI3K inhibitor, selectively targets FAP-expressing human idiopathic pulmonary fibrosis (IPF) cells. It effectively inhibits collagen synthesis and reduces collage... | |||
T35852 | FAPI-34 | ||
FAPI-34, a fibroblast-activating protein (FAP) inhibitor, boasts advantageous pharmacokinetic and biochemical attributes. | |||
T69660 | NOTA-FAPI-4 | ||
NOTA-FAPI-4 is an analogue of FAPI-4 and a fibroblast activation protein (FAP) inhibitor. NOTA-FAPI-4 is useful in the diagnosis or treatment of a disease characterized by overexpression of fibroblast activation protein... | |||
T82416 | FAPI-2 TFA | ||
FAPI-2 TFA is a fibroblast activation protein (FAP) inhibitor, potentially applicable in cancer research. [1] | |||
T11263 | FAPI-2 | Others | |
Fapi-2 is a fibroblast activated protein (FAP) inhibitor used in cancer research. | |||
T79917 | FAP-IN-2 | ||
FAP-IN-2 is a 99mTc-labeled, isonitrile-containing derivative of a fibroblast activation protein (FAPI) inhibitor suitable for tumor imaging [1]. | |||
T69603 | BR103354 | ||
BR103354 is a novel fibroblast activation protein (FAP) inhibitor with anti-diabetic and anti-steatotic effects. BR103354 inhibited FAP with an IC50 value of 14 nM, showing high selectivity against dipeptidyl peptidase (... | |||
T78179 | NH2-UAMC1110 TFA | ||
NH2-UAMC1110 TFA, a derivative of the fibroblast activation protein (FAP) inhibitor UAMC1110, serves as a precursor in the formation of FAPI-QS, a chelating agent crucial for creating radiotracers with high tumor selecti... | |||
T37861 | Talabostat | ||
Talabostat (PT100, Val-boroPro) is a potent, nonselective and orally available dipeptidyl peptidase IV (DPP-IV) inhibitor with a Ki of 0.18 nM. Talabostat is a nonselective DPP-IV inhibitor, inhibiting DPP8/9, FAP, DPP2 ... |